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Chemical structure of CAS 17692-51-2

Metergoline

In Stock•Starting at $239 for 50 mg
CAS No.17692-51-2
MDL No.N/A
MFC25H29N3O2
MW403.50
InChI KeyWZHJKEUHNJHDLS-QTGUNEKASA-N

Pricing & Availability

Pack SizePurityPriceAvailabilityAction
50 mgTo Be Confirmed$239In Stock
100 mgTo Be Confirmed$363In Stock
Custom synthesis and bulk supply options are available upon request.

Product Information

Metergoline is an ergoline alkaloid and carbamate ester, specifically the N-benzyloxycarbonyl derivative of lysergamine. It acts as a 5-HT2, 5-HT1, and 5-HT1D receptor antagonist, with moderate affinity for 5-HT6 and high affinity for 5-HT7. It functions as a serotonergic antagonist, dopamine agonist, and geroprotector.

CAS No.17692-51-2
Product NameMetergoline
IrritantIrritant
Signal Word:Warning
HCode:H302-H312-H332
PCode:P261-P264-P270-P271-P280-P301+P317-P302+P352-P304+P340-P317-P321-P330-P362+P364-P501

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Studies related to this compound and its mechanism of action

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Naunyn-Schmiedeberg's archives of pharmacology • Vol. 363, Issue 2 • 2001
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A role for serotonin in lipopolysaccharide-induced anorexia in rats.

Pharmacology, biochemistry, and behavior • Vol. 68, Issue 2 • 2001
PMID: 11267641DOI: 10.1016/s0091-3057(00)00463-9

Discriminative stimulus properties of indorenate, a 5-HT1A, 5-HT1B and 5-HT2C agonist: a study in rats.

Journal of psychopharmacology (Oxford, England) • Vol. 15, Issue 1 • 2001
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Documentation

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