Discovery of phosphoric acid mono-{2-[(E/Z)-4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-benzoylimino]-thiazol-3-ylmethyl} ester (Lu AA47070): a phosphonooxymethylene prodrug of a potent and selective hA(2A) receptor antagonist.
Journal of medicinal chemistry • Vol. 54, Issue 3 • 2011
Recent developments in adenosine receptor ligands and their potential as novel drugs.
Biochimica et biophysica acta • Vol. 1808, Issue 5 • 2011
Preladenant, a selective A(2A) receptor antagonist, is active in primate models of movement disorders.
Experimental neurology • Vol. 225, Issue 2 • 2010
Characterization of major degradation products of an adenosine A2A receptor antagonist under stressed conditions by LC-MS and FT tandem MS analysis.
Journal of mass spectrometry : JMS • Vol. 45, Issue 2 • 2010