Product Information

CAS No.	377727-87-2
Product Name	Preladenant

Biological Targets

ADORA2A

Associated Conditions

neoplasm·Parkinson disease·liver disease

* The information provided here is compiled from public sources and is for reference only.

Studies related to this compound and its mechanism of action

Discovery of phosphoric acid mono-{2-[(E/Z)-4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-benzoylimino]-thiazol-3-ylmethyl} ester (Lu AA47070): a phosphonooxymethylene prodrug of a potent and selective hA(2A) receptor antagonist.

Journal of medicinal chemistry • Vol. 54, Issue 3 • 2011

PMID: 21210664 DOI: 10.1021/jm1008659

Recent developments in adenosine receptor ligands and their potential as novel drugs.

Biochimica et biophysica acta • Vol. 1808, Issue 5 • 2011

PMID: 21185259 PMC: PMC3437328 DOI: 10.1016/j.bbamem.2010.12.017

Preladenant, a selective A(2A) receptor antagonist, is active in primate models of movement disorders.

Experimental neurology • Vol. 225, Issue 2 • 2010

PMID: 20655910 DOI: 10.1016/j.expneurol.2010.07.011

Characterization of major degradation products of an adenosine A2A receptor antagonist under stressed conditions by LC-MS and FT tandem MS analysis.

Journal of mass spectrometry : JMS • Vol. 45, Issue 2 • 2010

PMID: 19911413 DOI: 10.1002/jms.1695

Preladenant

CAS No.	377727-87-2
MDL No.	MFCD17167056
MF	C₂₅H₂₉N₉O₃
MW	503.60
InChI Key	DTYWJKSSUANMHD-UHFFFAOYSA-N

CUSTOM SYNTHESIS PRECLINICAL SUPPORT

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Custom synthesis and bulk supply options are available upon request.

Product Information

CAS No.	377727-87-2
Product Name	Preladenant

Biological Targets

ADORA2A

Associated Conditions

neoplasm·Parkinson disease·liver disease

* The information provided here is compiled from public sources and is for reference only.

Preladenant

Pricing & Availability

Product Information

Biological Profile

Safety Information

Properties

Biological Targets

Associated Conditions

Preladenant

Pricing & Availability

Product Information

Biological Profile

Safety Information

Properties

Biological Targets

Associated Conditions

Documentation

Preladenant

Pricing & Availability

Product Information

Biological Profile

Safety Information

Properties

Biological Targets

Associated Conditions

Related Articles

Discovery of phosphoric acid mono-{2-[(E/Z)-4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-benzoylimino]-thiazol-3-ylmethyl} ester (Lu AA47070): a phosphonooxymethylene prodrug of a potent and selective hA(2A) receptor antagonist.

Recent developments in adenosine receptor ligands and their potential as novel drugs.

Preladenant, a selective A(2A) receptor antagonist, is active in primate models of movement disorders.

Characterization of major degradation products of an adenosine A2A receptor antagonist under stressed conditions by LC-MS and FT tandem MS analysis.

Similar Products

Sch 58261

Preladenant

Pricing & Availability

Product Information

Biological Profile

Safety Information

Properties

Biological Targets

Associated Conditions

Related Articles

Discovery of phosphoric acid mono-{2-[(E/Z)-4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-benzoylimino]-thiazol-3-ylmethyl} ester (Lu AA47070): a phosphonooxymethylene prodrug of a potent and selective hA(2A) receptor antagonist.

Recent developments in adenosine receptor ligands and their potential as novel drugs.

Preladenant, a selective A(2A) receptor antagonist, is active in primate models of movement disorders.

Characterization of major degradation products of an adenosine A2A receptor antagonist under stressed conditions by LC-MS and FT tandem MS analysis.

Similar Products

Sch 58261

Documentation