Gsk2816126
| CAS No. | 1346574-57-9 |
|---|---|
| MDL No. | MFCD23381067 |
| MF | C31H38N6O2 |
| MW | 526.70 |
| InChI Key | FKSFKBQGSFSOSM-QFIPXVFZSA-N |
Pricing & Availability
| Pack Size | Purity | Price | Availability | Action |
|---|---|---|---|---|
| - | - | On Request | On Request | |
| Custom synthesis and bulk supply options are available upon request. | ||||
Product Information
GSK126 is a methylindole with substituents at positions 1, 3, 4, and 6: (2S)-butan-2-yl, methyl, N-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl]acetamide, and 6-(piperazin-1-yl)pyridin-3-yl groups. It is a potent and highly selective inhibitor of EZH2 methyltransferase (IC50 = 9.9 nM), acting as a neuroprotective, antiatherosclerotic, antineoplastic, anti-obesity, angiogenesis inhibitor, and EC 2.1.1.43 inhibitor. It belongs to pyridines, secondary carboxamides, pyridones, N-arylpiperazines, and methylindoles.
| CAS No. | 1346574-57-9 |
|---|---|
| Product Name | Gsk2816126 |
Biological Targets
EZH2
Associated Conditions
neoplasm·cancer
* The information provided here is compiled from public sources and is for reference only.
