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Chemical structure of CAS 1207253-08-4

Mk-1064

CAS No.1207253-08-4
MDL No.MFCD28502027
MFC24H20ClN5O3
MW461.90
InChI KeyCKTWQGHVNRYNCM-UHFFFAOYSA-N

Pricing & Availability

Pack SizePurityPriceAvailabilityAction
- -On RequestOn Request
Custom synthesis and bulk supply options are available upon request.

Product Information

CAS No.1207253-08-4
Product NameMk-1064
Health HazardHealth Hazard
Signal Word:Warning
HCode:H371-H373
PCode:P260-P264-P270-P308+P316-P319-P405-P501

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Scientific reports • Vol. 12, Issue 1 • 2022
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Orexin 2 Receptor Antagonism is Sufficient to Promote NREM and REM Sleep from Mouse to Man.

Scientific reports • Vol. 6 • 2016
PMID: 27256922PMC: PMC4891657DOI: 10.1038/srep27147

Discovery of 5''-chloro-N-[(5,6-dimethoxypyridin-2-yl)methyl]-2,2':5',3''-terpyridine-3'-carboxamide (MK-1064): a selective orexin 2 receptor antagonist (2-SORA) for the treatment of insomnia.

ChemMedChem • Vol. 9, Issue 2 • 2014
PMID: 24376006DOI: 10.1002/cmdc.201300447

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