Asp-3026
| CAS No. | 1097917-15-1 |
|---|---|
| MDL No. | MFCD21609265 |
| MF | C29H40N8O3S |
| MW | 580.70 |
| InChI Key | MGGBYMDAPCCKCT-UHFFFAOYSA-N |
Pricing & Availability
| Pack Size | Purity | Price | Availability | Action |
|---|---|---|---|---|
| - | - | On Request | On Request | |
| Custom synthesis and bulk supply options are available upon request. | ||||
Product Information
ASP-3026 is a diamino-1,3,5-triazine with 1,3,5-triazine-2,4-diamine core, where the amino groups at positions 2 and 4 are substituted with 2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl and 2-(propan-2-ylsulfonyl)phenyl groups, respectively. It is a potent inhibitor of ALK, Ack, and ROS1 (IC50: 3.5, 5.8, and 8.9 nM) and exhibits anti-cancer properties. It functions as an antineoplastic agent, apoptosis inducer, EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor, antimalarial, and EC 6.1.1.6 (lysine--tRNA ligase) inhibitor. It is classified as a secondary amino compound, monomethoxybenzene, N-methylpiperazine, aromatic amine, diamino-1,3,5-triazine, piperidine, and sulfone.
| CAS No. | 1097917-15-1 |
|---|---|
| Product Name | Asp-3026 |
Biological Targets
ALK
Associated Conditions
cancer·neoplasm of mature B-cells·neoplasm
* The information provided here is compiled from public sources and is for reference only.
