Effect of FAK inhibitor VS-6063 (defactinib) on docetaxel efficacy in prostate cancer.
The Prostate • Vol. 78, Issue 4 • 2018
The target landscape of clinical kinase drugs.
Science (New York, N.Y.) • Vol. 358, Issue 6367 • 2017
A first-in-Asian phase 1 study to evaluate safety, pharmacokinetics and clinical activity of VS-6063, a focal adhesion kinase (FAK) inhibitor in Japanese patients with advanced solid tumors.
Cancer chemotherapy and pharmacology • Vol. 77, Issue 5 • 2016
A phase I study of VS-6063, a second-generation focal adhesion kinase inhibitor, in patients with advanced solid tumors.
Investigational new drugs • Vol. 33, Issue 5 • 2015