PF-3758309
| CAS No. | 898044-15-0 |
|---|---|
| MDL No. | MFCD18633226 |
| MF | C25H30N8OS |
| MW | 490.60 |
| InChI Key | AYCPARAPKDAOEN-LJQANCHMSA-N |
Pricing & Availability
| Pack Size | Purity | Price | Availability | Action |
|---|---|---|---|---|
| - | - | On Request | On Request | |
| Custom synthesis and bulk supply options are available upon request. | ||||
Product Information
PF-3758309 is a thienopyrimidine containing a thieno[3,2-d]pyrimidine core substituted at positions 2 and 4 with a methyl group and a (5-{[(1S)-2-(dimethylamino)-1-phenylethyl]carbamoyl}-6,6-dimethyl-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)amino group, respectively. It is a potent PAK4 inhibitor that suppresses the growth of multiple human tumor xenografts. It functions as an EC 2.7.11.1 (non-specific serine/threonine protein kinase) inhibitor, an apoptosis inducer, and an antineoplastic agent. It is classified as a thienopyrimidine, pyrrolopyrazole, benzene derivative, urea, secondary amino compound, and tertiary amino compound.
| CAS No. | 898044-15-0 |
|---|---|
| Product Name | PF-3758309 |
Biological Targets
PAK4
Associated Conditions
neoplasm
* The information provided here is compiled from public sources and is for reference only.
