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Chemical structure of CAS 57717-80-3

CGP7930

CAS No.57717-80-3
MDL No.MFCD04040028
MFC19H32O2
MW292.50
InChI KeyXLWJPQQFJNGUPA-UHFFFAOYSA-N
CUSTOM SYNTHESISPRECLINICAL SUPPORT

Pricing & Availability

Pack SizePurityPriceAvailabilityAction
- -On RequestOn Request
Custom synthesis and bulk supply options are available upon request.

Product Information

2,6-Ditert-butyl-4-(3-hydroxy-2,2-dimethylpropyl)phenol is an alkylbenzene.

CAS No.57717-80-3
Product NameCGP7930
Heavy Atom Count21Rotatable Bond Count3
Atom Stereo Count0Bond Stereo Count0
HBA2HBD2
TPSA40.460 ŲCharge0
Exact Mass292.24023Complexity464.27
pKa8.400XLogP4.548

Related Articles

Studies related to this compound and its mechanism of action

Effects of GABA(B) receptor agents on cocaine priming, discrete contextual cue and food induced relapses.

European journal of pharmacology • Vol. 571, Issue 2-3 • 2007
PMID: 17610868DOI: 10.1016/j.ejphar.2007.05.069

CGP7930: a positive allosteric modulator of the GABAB receptor.

CNS drug reviews • Vol. 13, Issue 3 • 2007
PMID: 17894647PMC: PMC6494120DOI: 10.1111/j.1527-3458.2007.00021.x

Differential modulation by the GABAB receptor allosteric potentiator 2,6-di-tert-butyl-4-(3-hydroxy-2,2-dimethylpropyl)-phenol (CGP7930) of synaptic transmission in the rat hippocampal CA1 area.

The Journal of pharmacology and experimental therapeutics • Vol. 317, Issue 3 • 2006
PMID: 16507713DOI: 10.1124/jpet.105.099176

Reducing effect of the positive allosteric modulators of the GABA(B) receptor, CGP7930 and GS39783, on alcohol intake in alcohol-preferring rats.

European journal of pharmacology • Vol. 525, Issue 1-3 • 2005
PMID: 16289452DOI: 10.1016/j.ejphar.2005.10.005

Documentation

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