Acylated Gly-(2-cyano)pyrrolidines as inhibitors of fibroblast activation protein (FAP) and the issue of FAP/prolyl oligopeptidase (PREP)-selectivity.
Bioorganic & medicinal chemistry letters • Vol. 22, Issue 10 • 2012
Synthesis of novel aza-analogues of tiazofurin with 2-[5,5-bis(hydroxymethyl)pyrrolidin-2-yl] framework as sugar mimic.
Nucleosides, nucleotides & nucleic acids • Vol. 31, Issue 1 • 2012
Synthesis and evaluation of structurally constrained imidazolidin derivatives as potent dipeptidyl peptidase IV inhibitors.
European journal of medicinal chemistry • Vol. 44, Issue 8 • 2009
Discovery of conformationally rigid 3-azabicyclo[3.1.0]hexane-derived dipeptidyl peptidase-IV inhibitors.
Bioorganic & medicinal chemistry letters • Vol. 18, Issue 14 • 2008