Potency of nonnucleoside reverse transcriptase inhibitors (NNRTIs) used in combination with other human immunodeficiency virus NNRTIs, NRTIs, or protease inhibitors.
Antimicrobial agents and chemotherapy • Vol. 46, Issue 6 • 2002
3,3a-Dihydropyrano[4,3,2-de]quinazolin-2(1H)-ones are potent non-nucleoside reverse transcriptase inhibitors.
Bioorganic & medicinal chemistry letters • Vol. 11, Issue 2 • 2001
Trifluoromethyl-containing 3-alkoxymethyl- and 3-aryloxymethyl-2-pyridinones are potent inhibitors of HIV-1 non-nucleoside reverse transcriptase.
Bioorganic & medicinal chemistry letters • Vol. 11, Issue 3 • 2001
4,1-Benzoxazepinone analogues of efavirenz (Sustiva) as HIV-1 reverse transcriptase inhibitors.
Bioorganic & medicinal chemistry letters • Vol. 11, Issue 11 • 2001