Identification of (R)-N-((4-Methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)ethyl)-1H-indole-3-carboxamide (CPI-1205), a Potent and Selective Inhibitor of Histone Methyltransferase EZH2, Suitable for Phase I Clinical Trials for B-Cell Lymphomas.
Journal of medicinal chemistry • Vol. 59, Issue 21 • 2016
Identification of EZH2 and EZH1 small molecule inhibitors with selective impact on diffuse large B cell lymphoma cell growth.
Chemistry & biology • Vol. 20, Issue 11 • 2013
Resistance to freezing by Antarctic fauna: supercooling and osmoregulation.
Comparative biochemistry and physiology. A, Comparative physiology • Vol. 54, Issue 3 • 1976
