IGF2BP1 induces neuroblastoma via a druggable feedforward loop with MYCN promoting 17q oncogene expression.
Molecular cancer • Vol. 22, Issue 1 • 2023
Comprehensive transcriptome profiling of BET inhibitor-treated HepG2 cells.
PloS one • Vol. 17, Issue 4 • 2022
Superior efficacy of cotreatment with BET protein inhibitor and BCL2 or MCL1 inhibitor against AML blast progenitor cells.
Blood cancer journal • Vol. 9, Issue 2 • 2019
Discovery of N-(4-(2,4-Difluorophenoxy)-3-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)phenyl)ethanesulfonamide (ABBV-075/Mivebresib), a Potent and Orally Available Bromodomain and Extraterminal Domain (BET) Family Bromodomain Inhibitor.
Journal of medicinal chemistry • Vol. 60, Issue 20 • 2017