Development of a potent benzonitrile-based inhibitor of glutaminyl-peptide cyclotransferase-like protein (QPCTL) with antitumor efficacy.
Signal transduction and targeted therapy • Vol. 8, Issue 1 • 2023
Development and evolution of human glutaminyl cyclase inhibitors (QCIs): an alternative promising approach for disease-modifying treatment of Alzheimer's disease.
Frontiers in aging neuroscience • Vol. 15 • 2023
Glutaminyl cyclases, the potential targets of cancer and neurodegenerative diseases.
European journal of pharmacology • Vol. 931 • 2022
Glutaminyl Cyclase Inhibitor PQ912 Improves Cognition in Mouse Models of Alzheimer's Disease-Studies on Relation to Effective Target Occupancy.
The Journal of pharmacology and experimental therapeutics • Vol. 362, Issue 1 • 2017