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Chemical structure of CAS 1001389-72-5

Gsk-1482160

CAS No.1001389-72-5
MDL No.MFCD30532733
MFC14H14ClF3N2O2
MW334.72
InChI KeyBJEMSIVBBUBXMZ-JTQLQIEISA-N
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Product Information

CAS No.1001389-72-5
Product NameGsk-1482160

Biological Targets

P2RX7

Associated Conditions

Pain
* The information provided here is compiled from public sources and is for reference only.

Related Articles

Studies related to this compound and its mechanism of action

The IUPHAR Guide to Immunopharmacology: connecting immunology and pharmacology.

Immunology • Vol. 160, Issue 1 • 2020
PMID: 32020584PMC: PMC7160657DOI: 10.1111/imm.13175

Pyroglutamide-Based P2X7 Receptor Antagonists Targeting Inflammatory Bowel Disease.

Journal of medicinal chemistry • Vol. 63, Issue 5 • 2020
PMID: 31525963DOI: 10.1021/acs.jmedchem.9b00584

Characterization of C-GSK1482160 for Targeting the P2X7 Receptor as a Biomarker for Neuroinflammation.

Journal of nuclear medicine : official publication, Society of Nuclear Medicine • Vol. 58, Issue 3 • 2017
PMID: 27765863DOI: 10.2967/jnumed.116.181354

Discovery and structure-activity relationships of a series of pyroglutamic acid amide antagonists of the P2X7 receptor.

Bioorganic & medicinal chemistry letters • Vol. 20, Issue 17 • 2010
PMID: 20673717DOI: 10.1016/j.bmcl.2010.07.033

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